CPI-360 CellCPI 360 is a potent, selective,and SAM competitive EZH1 inhibitor with IC50 of 102. 3 nM, >100 fold selectivity over other methyltransferases.
Cholestyramine resin is a strongly basic anion exchange resin which can exchange its chloride anions with anionic bile acids in the gastrointestinal tract and bind them strongly in the resin matrix
and also a DNA/RNA synthesis inhibitor by intercalating into DNA and interacts with topoisomerase II
kinase activation
Pyridoxine HCl is a form of vitamin B6
acts as a selective inhibitor for neuronal nitric oxide synthase showing a 10-fold selectivity for neuronal NOS
Alcaftadine is also an antagonist for H2 and H4 receptors with no affinity for the H3 receptor
a novel sphingosine-competitive inhibitor of SphK1
Anthraquinones are the main active constituents in herbs often used to relieve constipation
Streptozotocin is a glucosamine-nitrosourea derivative
Rimantadine is an RNA synthesis inhibitor that is used as an antiviral agent in the prophylaxis and treatment of influenza
competitively inhibiting the interaction between gp120 and CD4
GGTI 298 is a geranylgeranyltransferase I inhibitor with ability to arrest human tumor cells in the G1 phase of the cell cycle and induce apoptosis
